Acne Treatment with Prescription Topicals

In the previous post we have discussed the the three over the counter acne treatments most commonly used. These are salicylic acid, sulfur, and benzoyl peroxide. Other topical acne treatment require a doctor's prescription due to potential side effects. They are used for mild-to-moderate cases of acne and many are chemically related to Vitamin A. They are:

Azelaic Acid

  • Azelaic acid is an organic compound naturally found in wheat, barley, and rye.
  • It is effective for mild and moderate outbreaks of acne by killing bacteria
  • Also acts as a keratolytic agent
  • Does not work quite well for acne that does not involve bacterial infection
  • Available as cream at 20% concentration
  • Can irritate the skin and cause hypopigmentation
  • Must be prescribed by a health care provider
  • Applied twice a day
  • Works as well as other agents (tretinoin, benzoyl peroxide)
  • Takes 1-2 months to start clearing your acne
  • Active ingredient in Azelex®, Finevin®, and Finacea®

Tretinoin

  • Tretinoin is the best known among the retinoids, a class of compounds chemically related to Vitamin A
  • Works by increasing skin cell turnover, which promotes the removal and prevention of blackheads and whiteheads
  • Available on prescription as cream (from 0.025% to 0.1%), as gel (0.01% to 0.05%), and as liquid (0.05%)
  • Benzoyl peroxide deactivates tretinoin; therefore, these two cannot be applied together at the same time
  • May seem to make acne worse at the start but it must be given time to work, 2-3 months at best
  • Can improve wrinkles and fine lines but makes the skin more susceptible to drying, redness, and sunburn; do not use more than the recommended amount to minimize side effects
  • Available as generic. Its brand names are Retin-A®, Avita®, and Renova®

Adapalene

  • Adapelene is a third-generation retinoid, just like tretinoin, but is newer and just as effective
  • Better tolerated or has fewer side effects than tretinoin
  • May be applied together with benzoyl peroxide
  • Available as the brand name Differin®, in a gel or cream form at 0.1% strength

Tazarotene

  • Tazarotene is another retinoid and like adapelene is also newer than tretinoin
  • A head-to-head comparison study conducted by Dr. Leyden of the University of Pennsylvania showed that Tazarotene was more effective than tretinoin
  • Commonly sold as a gel at 0.05% and 0.1% concentrations
  • More expensive compared to the other retinoids
  • Causes the same side effects as tretinoin
  • Marketed as Tazorac®, Avage®, and Zorac®

Next: Acne Treatment with Topical Antibiotics